Synthesis and multitarget inhibitory effect of indole-based ethyl cinnamate derivatives against SARS-CoV-2 Mpro and cathepsins for broad-spectrum anti-coronavirus activity

Bioorganic and Medicinal Chemistry 2025, DOI: 10.1016/j.bmc.2025.118258

Andrea Citarella, Giulia Sibille, Davide Moi, Alessandro Dimasi, Tommaso Braga, Lorenzo Dal Col, Lorenzo Ruberto, Stefano Pieraccini, Maurizio Sironi, Nicola Micale, Tanja Schirmeister, Valerio Fasano, Alessandra Silvani, Clelia Giannini, Giorgio Gribaudo, Daniele Passarella