Recent Publications – Page 3

A Green Approach to Nucleophilic Aromatic Substitutions of Nicotinic Esters in Cyrene

European Journal of Organic Chemistry 2024, e202301305

Andrea Citarella,* Miriam Cavinato, Arianna Amenta, Marco Nardini, Alessandra Silvani, Daniele Passarella and Valerio Fasano*

Targeting Ovarian Cancer with chalcone Derivatives: Cytotoxicity and Apoptosis Induction in HGSOC Cells

Molecules 2023, 28 (23), 7777

Elif Merve Aydin,Idil Su Canıtez, Eleonora Colombo, Salvatore Princiotto, Daniele Passarella, Sabrina Dallavalle, Michael S. Christodoulou and Irem Durmaz Sahin

Modular Symmetric Ligands for Selective Recognition of Cancer-Relevant G-Quadruplexes

Chiara Platella, Andrea Citarella, Marco Manenti, Guglielmo Spinelli, Rosa Gaglione, Angela Arciello, Claudia Riccardi, Domenica Musumeci, Daniela Montesarchio, Clelia Giannini, Alessandra Silvani

Journal of Molecular Structure, 2024, 5, 137114

https://doi.org/10.1016/j.molstruc.2023.137114

Recent Advances in SARS-CoV-2 Main Protease Inhibitors: From Nirmatrelvir to Future Perspectives

A. Citarella, A. Dimasi, D. Moi, D. Passarella, A. Scala, A. Piperno, N. Micale

Biomolecules. (2023)

10.3390/biom13091339

Recent advances in the development of CB1R selective probes

A. Amenta, D. Caprioglio, A. Minassi, L. Panza, D. Passarella, V. Fasano, D. Imperio

Front. Nat. Prod. (2023)

10.3389/fntpr.2023.1196321

Synthesis and Preliminary Characterization of Putative Anle138b-Centered PROTACs against α-Synuclein Aggregation

M. Pedrini, A. Iannielli, L. Meneghelli, D. Passarella, V. Broccoli, P. Seneci

Pharmaceutics (2023)

10.3390/pharmaceutics15051467

2-Hydroxyoleic Acid as a Self-Assembly Inducer for Anti-Cancer Drug-Centered Nanoparticles

A. I. Antoniou, G. Nordio, M. L. Di Paolo, E. Colombo, B. Gaffuri, L. Polito, A. Amenta, P. Seneci, L. Dalla Via, D. Perdicchia, D. Passarella

Pharmaceutics (2023)

10.3390/ph16050722

Dual targeted 2-Benzylideneindanone pendant hydroxamic acid group exhibits selective HDAC6 inhibition along with tubulin stabilization effect

K. Kumar, R. Das, B. Thapa, B. Rakhecha, S. Srivastav, K. Savita, M. Israr, D. Chanda, D. Banerjee, K. Shanker, D.U. Bawankule, B. Santini, M. L. Di Paolo, L. Dalla Via, D. Passarella, A. Singh Negi

Bioorg. Med. Chem. (2023)

10.1016/j.bmc.2023.117300

Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses

A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella

Org. Biomol. Chem. (2023)

10.1039/D3OB00381G

Late-Stage Functionalisation of Pyridine-Containing Bioactive Molecules: Recent Strategies and Perspectives

M. Failla; G. W. Lombardo; P. Orlando; D. Fiorito; E. Bombonato; P. Ronchi; D. Passarella; V. Fasano

EurJOC (2023)

10.1002/ejoc.202300074

Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro

A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, D. Passarella, C. Giannini

Molecules (2023)

10.3390/molecules28020514

Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics

Z. Boiarska, H. Pérez-Peña, A.-C. Abel, P. Marzullo, B. Álvarez-Bernad, F. Bonato, B. Santini, D. Horvath, D. Lucena-Agell, F. Vasile, M. Sironi, J. F. Díaz, A. E. Prota, S. Pieraccini, D. Passarella

Chem. Eur. J. (2022)

10.1002/chem.202203431