Recent advances in the development of CB1R selective probes
A. Amenta, D. Caprioglio, A. Minassi, L. Panza, D. Passarella, V. Fasano, D. Imperio
Front. Nat. Prod. (2023)
Synthesis and Preliminary Characterization of Putative Anle138b-Centered PROTACs against α-Synuclein Aggregation
M. Pedrini, A. Iannielli, L. Meneghelli, D. Passarella, V. Broccoli, P. Seneci
Pharmaceutics (2023)
2-Hydroxyoleic Acid as a Self-Assembly Inducer for Anti-Cancer Drug-Centered Nanoparticles
A. I. Antoniou, G. Nordio, M. L. Di Paolo, E. Colombo, B. Gaffuri, L. Polito, A. Amenta, P. Seneci, L. Dalla Via, D. Perdicchia, D. Passarella
Pharmaceutics (2023)
Dual targeted 2-Benzylideneindanone pendant hydroxamic acid group exhibits selective HDAC6 inhibition along with tubulin stabilization effect
K. Kumar, R. Das, B. Thapa, B. Rakhecha, S. Srivastav, K. Savita, M. Israr, D. Chanda, D. Banerjee, K. Shanker, D.U. Bawankule, B. Santini, M. L. Di Paolo, L. Dalla Via, D. Passarella, A. Singh Negi
Bioorg. Med. Chem. (2023)
Synthesis of SARS-CoV-2 Mpro Inhibitors bearing a Cinnamic Ester Warhead with In Vitro Activity against Human Coronaviruses
A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, A. Dimasi, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, C. Giannini, D. Passarella
Org. Biomol. Chem. (2023)
Late-Stage Functionalisation of Pyridine-Containing Bioactive Molecules: Recent Strategies and Perspectives
M. Failla; G. W. Lombardo; P. Orlando; D. Fiorito; E. Bombonato; P. Ronchi; D. Passarella; V. Fasano
EurJOC (2023)
Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 Mpro
A. Citarella, D. Moi, M. Pedrini, H. Pérez-Peña, S. Pieraccini, C. Stagno, N. Micale, T. Schirmeister, G. Sibille, G. Gribaudo, A. Silvani, D. Passarella, C. Giannini
Molecules (2023)
Maytansinol Functionalization: Towards Useful Probes for Studying Microtubule Dynamics
Z. Boiarska, H. Pérez-Peña, A.-C. Abel, P. Marzullo, B. Álvarez-Bernad, F. Bonato, B. Santini, D. Horvath, D. Lucena-Agell, F. Vasile, M. Sironi, J. F. Díaz, A. E. Prota, S. Pieraccini, D. Passarella
Chem. Eur. J. (2022)
Cyrene: A Green Solvent for the Synthesis of Bioactive Molecules and Functional Biomaterials
A. Citarella, A. Amenta, D. Passarella, N. Micale
Int. J. Mol. Sci. (2022)
Folic acid functionalization for targeting self-assembled paclitaxel-based nanoparticles
E. Colombo, D.A. Coppini, S. Maculan, P. Seneci, B. Santini, F. Testa, L. Salvioni, G. Vanacore, M. Colombo, D. Passarella
RSC Advances (2022)
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors
A. Tinivella, J. C. Nwachukwu, A. Angeli, F. Foschi, A. L. Benatti, L. Pinzi, T. Izard, M. Ferraroni, R. Erumbi, M. S. Christodoulou, D. Passarella, C. T. Supuran, K. W. Nettles, G. Rastelli
European Journal of Medicinal Chemistry (2022)
Dual-functionalized liposomes for selective delivery of poorly soluble drugs to inflamed brain regions
S. Giofrè, A. Renda, S. Sesana, B. Formicola, B. Vergani, B.E. Leone, V. Denti, G. Paglia, S. Groppuso, V. Romeo, L. Muzio, A. Balboni, A. Menegon, A. Antoniou, A. Amenta, D. Passarella, P. Seneci, S. Pellegrino, F. Re
Pharmaceutics (2022)