Synthesis and biological evaluation of novel tamoxifen analogues
M. S. Christodoulou, N. Fokialakis, D. Passarella, A. N. García-Argáez, O. M. Gia, I. Pongratz, L. Dalla Via, S. A. Haroutounian
Bioorg. Med. Chem. (2013), 21, 4120-4131
9-Fluorenone-2-carboxylic acid as scaffold for new tubulin interacting compounds
F. Calogero, S. Borrelli, G. Speciale, M. S. Christodoulou, D. Cartelli, D. Ballinari, F. Sola , C. Albanese, A. Ciavolella, D. Passarella, G. Cappelletti, S. Pieraccini, M. Sironi
ChemPlusChem (2013), 78, 663-669
DOI: 10.1002/cplu.201300036
Microtubule alterations occur early in experimental parkinsonism and the microtubule stabilizer epothilone D is neuroprotective
D. Cartelli, F. Casagrande, C. L. Busceti, D. Bucci, G. Molinaro, A. Traficante, D. Passarella, E. Giavini, G. Battaglia, G. Cappelletti
Scientific Reports 2013, 3: 1837
DOI: 10.1038/srep01837
Probing the Binding Site of Abl Tyrosine Kinase Using in Situ Click Chemistry
C. Peruzzotti, S. Borrelli, M. Ventura, R. Pantano, G. Fumagalli, M. S. Christodoulou, D. Monticelli, M. Luzzani, A. L. Fallacara, C. Tintori, M. Botta, D. Passarella
ACS Med. Chem. Letters 2013, 4, 274-277
DOI: 10.1021/ml300394w
Preparation of Fluorescent Tubulin Binders
34. E. Riva, M. Mattarella, S. Borrelli, M. S. Christodoulou, D. Cartelli, M. Main, S. Faulkner, D. Sykes, G. Cappelletti, J. S. Snaith, D. Passarella
ChemPlusChem 2013, 3, 222
DOI: 10.1002/cplu.201200260
Cover 2013, 3, 201
Camptothecin-7-yl-methanthiole: Semisynthesis and Biological Evaluation
M. S. Christodoulou , F. Zunino, V. Zuco, S. Borrelli, D. Comi, G. Fontana, M. Martinelli, J. Lorens, L. Evensen, M. Sironi, S. Pieraccini, L. Dalla Via, O. M. Gia, D. Passarella
ChemMedChem (2012),7, 2134-2143
DOI: 10.1002/cmdc.201200322
Combined drug action of 2-phenylimidazo[2,1-b]benzothiazole derivatives on cancer cells according to their oncogenic molecular signatures
A. Furlan, B. Roux, F. Lamballe, F. Conti, N. Issaly, F. Dalan, J-F. Gullemot, S. Richelme, M. Contersin, J. Bosch, D. Passarella, O. Piccolo, R. Dono , F. Maina
PLOSEone 7 (10) , art. no. e46738
‘Click’synthesis of a triazole-based inhibitor of Met functions in cancer cells
F. Colombo, C. Tintori, A. Furlan, S. Borrelli, M. S. Christodoulou, R. Dono, F. Maina, M. Botta, M. Amat, J. Bosch, D. Passarella
Biorg.Med.ChemLett. (2012), 22, 4693 – 4696
Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signalling
A. Furlan, F. Colombo, A. Kover, N. Issaly, C. Tintori, L. Angeli, V. Leroux, S. Letard, M. Amat, Y. Asses, B. Maigret, P. Dubreuil, M. Botta, R. Dono, J. Bosch, O. Piccolo, D. Passarella, F. Maina
Eur.J.Med.Chem (2012), 47, 239-254
Chiral flavanones from Amygdalus lycioides Spach: structural elucidation and identification of TNFalpha inhibitors by bioactivity-guided fractionation
R. Gaggeri, D. Rossi, M.S. Christodoulou, D. Passarella, F. Leoni, O. Azzolina, S. Collina
Molecules, (2012), 17, 1665-1674
N-[2-Methyl-5-(triazol-1-yl)phenyl]pyrimidin-2-amine as a Scaffold for the Synthesis of Inhibitors of Bcr-Abl
F. Arioli, S. Borrelli, F. Colombo, F. Falchi, I. Filippi, E. Crespan, A. Naldini, G. Scalia, A. Silvani, G. Maga, F. Carraro, M. Botta, D. Passarella
ChemMedChem (2011), 6, 2009 – 2018
DOI: 10.1002/cmdc.201100304
Tubulin-guided dynamic combinatorial library of thiocolchicine-podophyllotoxin conjugates
G. Cappelletti, D. Cartelli, B. Peretto, M. Ventura, M. Riccioli, F. Colombo, J. S. Snaith, S. Borrelli, D. Passarella
Tetrahedron (2011), 67, 7354 – 7357
doi:10.1016/j.tet.2011.07.038